Amiloride HCl

Catalog No.: A10064

Na+ channel blocker

Amiloride HCl

Amiloride HCl Chemical Structure

CAS NO. 2016-88-8

Amiloride hydrochloride is a Na+ channel blocker, also inhibits TRPP3 channels and Na+/H+ exchanger (NHE).

Availability: In stock

Package Price Qty
200 mg
500 mg
10mM * 1mL in DMSO
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Yu Y, .et al. Expression, Localization and Functional Activity of the Major Na+/H+ Exchange Isoforms Expressed in the Intestinal Cell Line Caco-2BBe, Cell Physiol Biochem, 2019, 52(5):1017-1038 PMID: 30977986
  • Thomas D. Williams, .et al. The physiological regulation of macropinocytosis during Dictyostelium growth and development, J Cell Sci, 2018, Mar 15; 131(6): jcs213736 PMID: 29440238

Biological Activity

Amiloride hydrochloride is a Na+ channel blocker, also inhibits TRPP3 channels and Na+/H+ exchanger (NHE).
In vitro DMSO 49 mg/mL (184.15 mM)
Water 6 mg/mL (22.54 mM)
Ethanol 5 mg/mL (18.79 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 37.58 mL 187.9 mL 375.8 mL
0.5 mM 7.52 mL 37.58 mL 75.16 mL
1 mM 3.76 mL 18.79 mL 37.58 mL
5 mM 0.75 mL 3.76 mL 7.52 mL

*The above data is based on the productmolecular weight 266.1 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10064
Actions Blocker
CAS No. 2016-88-8
Formula C6H9Cl2N7O
M. Wt 266.1
Purity >98%
Synonyms MK 870, Midamor, Colectril, Amipramizide, Guanamprazine hydrochloride
SMILES C1(=C(N=C(C(=N1)Cl)N)N)C(=O)N=C(N)N.Cl

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
You may also be interested in the following product(s)
Keywords:buy Amiloride HCl | Amiloride HCl Supplier | purchase | cost | manufacturer | order | distributor | buy 2016-88-8 | 2016-88-8 Supplier | purchase 2016-88-8 | 2016-88-8 cost | 2016-88-8 manufacturer | order 2016-88-8 | 2016-88-8 distributor