Fig. 1 · Structure
Documents & Downloads
Anpirtoline
5-HT1B Receptor Agonist
Anpirtoline is a potent agonist of the 5-HT1B receptor, exhibiting a Ki of 28 nM for this target, alongside 150 nM for 5-HT1A and 1.49 μM for 5-HT2 receptors. This compound demonstrates notable serotonergic activity and has been linked to antinociceptive and antidepressant-like effects. Anpirtoline is primarily utilized in research to explore its potential therapeutic applications in mood disorders and pain management.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 98330-05-3 |
| Applications | 5-HT1B Receptor Agonist |
| Formula | C10H13ClN2S |
| Molecular Weight | 228.74 |
| Synonyms | D-16949 |
| SMILES | ClC1=NC(SC2CCNCC2)=CC=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.