Fig. 1 · Structure
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Antitrypanosomal agent 7
Antitrypanosomal Agent
Antitrypanosomal agent 7 is a potent inhibitor targeting Trypanosoma brucei, demonstrating superior efficacy compared to Nifurtimox, with an IC50 value of 0.71 μM. This compound exhibits favorable ADME properties and a strong affinity for DNA, selectively binding to AT-rich regions. Its bioactivity makes it a valuable tool for research applications focused on trypanosomiasis and drug development against parasitic diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2492436-38-9 |
| Applications | Antitrypanosomal Agent |
| Formula | C23H31Cl2N5O2 |
| Molecular Weight | 480.43 |
| SMILES | COC1=CC(C2=NC3=CC(C4=NCCN4)=CC=C3N2)=CC=C1OCCN(CC)CC.[H]Cl.[H]Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.