Fig. 1 · Structure
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Apelin-36(human)
APJ Agonist
Apelin-36 (human) is a potent agonist for the APJ receptor, demonstrating an EC50 of 20 nM. It exhibits high affinity for human APJ receptors expressed in HEK 293 cells, indicated by a pIC50 value of 8.61. Apelin-36 is primarily involved in cardiovascular and metabolic regulation and has also been shown to inhibit the entry of HIV-1 and HIV-2 into NP2/CD4 cells that express the APJ receptor, making it relevant in virology research.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 252642-12-9 |
| Applications | APJ Agonist |
| Formula | C184H297N69O43S |
| Molecular Weight | 4195.83 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.