Aprepitant-13C2,d2 (Major)

Catalog No.: A47267
Stable Isotope
Aprepitant-13C2,d2 (Major) is a stable isotope-labeled variant of Aprepitant, a selective and high-affinity antagonist of the neurokinin 1 receptor with a dissociation constant (Kd) of 86 pM. This reagent is primarily utilized in pharmacokinetic studies and metabolic research. The 13C labeling allows for precise tracing and quantification in complex biological systems, facilitating a deeper understanding of Aprepitant's biochemical interactions and tissue distribution.
Grouped product items
Size Price Stock Qty
1mg
$400.00
In stock
10mg
$3,175.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Nature Volume 622 Issue 7982 (2023)
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Nature volume 551, pages639-643 (2017)
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Biological Activity
DescriptionAprepitant-13C2,d2 (Major) is a stable isotope-labeled variant of Aprepitant, a selective and high-affinity antagonist of the neurokinin 1 receptor with a dissociation constant (Kd) of 86 pM. This reagent is primarily utilized in pharmacokinetic studies and metabolic research. The 13C labeling allows for precise tracing and quantification in complex biological systems, facilitating a deeper understanding of Aprepitant's biochemical interactions and tissue distribution.
Product Information
Catalog NumA47267
FormulaC2113C2H19D2F7N4O3
Molecular Weight538.42
CAS Number1217676-37-3
SMILESO=C1N[13C]([13CH2]N2CCO[C@@H]([C@@H]2C3=CC=C(C=C3)F)O[C@](C[2H])(C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)[2H])=NN1
SynonymsMK-0869--13C2,d2; MK-869-13C2,d2; L-754030--13C2,d2
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