Fig. 1 · Structure
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Asivatrep
Cat. No.
A68717
CAS
1005168-10-4
TRP Channel Antagonist
Asivatrep (PAC-14028) is a potent and selective antagonist of the transient receptor potential vanilloid type I (TRPV1) channel. This compound exhibits significant analgesic effects by blocking TRPV1, which is involved in the transmission of nociceptive signals. Asivatrep is primarily utilized in research related to pain management and neurobiology. Its selective inhibition offers a valuable tool for studying TRPV1-mediated pathways and their role in various physiological and pathological conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1005168-10-4 |
| Applications | TRP Channel Antagonist |
| Formula | C21H22F5N3O3S |
| Molecular Weight | 491.47 |
| Synonyms | PAC-14028 |
| SMILES | O=C(N[C@@H](C1=CC(F)=C(NS(=O)(C)=O)C(F)=C1)C)/C=C/C2=CC=C(C(F)(F)F)N=C2CCC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.