aTAG 2139

Name: aTAG 2139
Brand: Adooq Bioscience
SKU: A38361
Rating: 5 (288 reviews)

Catalog No.: A38361

MTH1 Degrader

aTAG 2139 is a selective degrader targeting MTH1 via an aTAG-based mechanism. It demonstrates biological activity with a DC50 value of 1.1 nM and a Ki value of 2.1 nM for MTH1 inhibition. This compound is suitable for studies investigating the role of MTH1 in various cellular processes and therapeutic applications in cancer research.

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Size	Price	Stock
1mg	$285.00	In stock
5mg	$870.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	aTAG 2139 is a selective degrader targeting MTH1 via an aTAG-based mechanism. It demonstrates biological activity with a DC50 value of 1.1 nM and a Ki value of 2.1 nM for MTH1 inhibition. This compound is suitable for studies investigating the role of MTH1 in various cellular processes and therapeutic applications in cancer research.

Product Information

Catalog Num	A38361
Formula	C42H38N8O8
Molecular Weight	782.80
CAS Number	2387510-81-6
SMILES	O=C(C1=CC=C(C2=CC=C3N=CC(C(NC)=O)=C(C3=C2)NC4=CC=CC=C4)C=N1)NCCCCNC(COC5=CC=CC(C(N6C7C(NC(CC7)=O)=O)=O)=C5C6=O)=O
Synonyms	CFT-2139

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