AZ6102

Catalog No.: A15873

TNKS1/2 inhibitor

AZ6102 Chemical Structure

CAS NO. 1645286-75-4

AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.

Availability: In stock

Package Price Qty
10 mg
$110.00
25 mg
$200.00
50 mg
$400.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.
Targets
TNKS1 TNKS2
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.34 mL 116.68 mL 233.36 mL
0.5 mM 4.67 mL 23.34 mL 46.67 mL
1 mM 2.33 mL 11.67 mL 23.34 mL
5 mM 0.47 mL 2.33 mL 4.67 mL

*The above data is based on the productmolecular weight 428.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15873
Actions Inhibitor
M. Wt 428.53
Formula C25H28N6O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1645286-75-4
Synonyms AZ-6102, AZ 6102
SMILES C[[email protected]]1CN(C2=NC=C(C3=CC=C(C4=NC(C(C=CN5C)=C5N4)=O)C=C3)C(C)=C2)C[[email protected]@H](C)N1

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