AZ6102

Catalog No.: A15873

TNKS1/2 inhibitor

AZ6102

AZ6102 Chemical Structure

CAS NO. 1645286-75-4

AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.

Availability: In stock

Package Price Qty
10 mg
$110.00
25 mg
$200.00
50 mg
$400.00
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Biological Activity

AZ6102 is a potent TNKS1/2 inhibitor that has 100-fold selectivity against other PARP family enzymes and shows IC50 of 5 nM for Wnt pathway inhibition in DLD-1 cells.
Targets
TNKS1 TNKS2
In vitro DMSO 83 mg/mL (193.68 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.34 mL 116.68 mL 233.36 mL
0.5 mM 4.67 mL 23.34 mL 46.67 mL
1 mM 2.33 mL 11.67 mL 23.34 mL
5 mM 0.47 mL 2.33 mL 4.67 mL

*The above data is based on the productmolecular weight 428.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15873
Actions Inhibitor
CAS No. 1645286-75-4
Formula C25H28N6O
M. Wt 428.53
Solubility DMSO
Purity >98%
Synonyms AZ-6102, AZ 6102
SMILES C[[email protected]]1CN(C2=NC=C(C3=CC=C(C4=NC(C(C=CN5C)=C5N4)=O)C=C3)C(C)=C2)C[[email protected]@H](C)N1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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