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β2AR/M-receptor agonist-1

Muscarinic Receptor Antagonist

β2AR/M-receptor agonist-1 is a dual-function compound acting as a muscarinic receptor antagonist and β2 adrenoceptor agonist. It exhibits a potent agonistic effect on the β2 adrenoceptor, with an EC50 value of 9.2 nM, and also demonstrates antagonistic activity against the muscarinic receptor, characterized by a Ki value of 30.2 nM. This compound is valuable for research applications involving modulation of adrenergic and muscarinic signaling pathways.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	2230520-62-2
Applications	Muscarinic Receptor Antagonist
Formula	C₄₃H₅₆BrN₃O₇
Molecular Weight	806.82
SMILES	O[C@@H](C1=C2C(NC(C=C2)=O)=C(C=C1)O)CNCCCOC(C=C3)=CC=C3OCCC[N+]45C[C@H](C(CC5)CC4)OC[C@@](C6CCCC6)(C7=CC=CC=C7)O.[Br-]

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.