BD-9136 is a potent and highly selective BRD4-targeting PROTAC degrader. It exhibits low-nanomolar degradation potency against BRD4, with over 1000-fold selectivity compared to BRD2 and BRD3. BD-9136 also demonstrates antitumor activity.
BD-9136 is a potent and highly selective BRD4-targeting PROTAC degrader. It exhibits low-nanomolar degradation potency against BRD4, with over 1000-fold selectivity compared to BRD2 and BRD3. BD-9136 also demonstrates antitumor activity.
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula: