bio-THZ1

Catalog No.: A18559

covalent CDK7 inhibitor

bio-THZ1

bio-THZ1 Chemical Structure

CAS NO. 1604811-14-4

bio-THZ1 is a biotinylated version of THZ1 and binds irreversibly to CDK7. THZ1 is a selective and potent covalent CDK7 inhibitor with an IC50 of 3.2 nM.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $350.00

Special Price $280.00

10 mg

Regular Price: $650.00

Special Price $520.00

50 mg

Regular Price: $2,000.00

Special Price $1,600.00

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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

bio-THZ1 is a biotinylated version of THZ1 and binds irreversibly to CDK7. THZ1 is a selective and potent covalent CDK7 inhibitor with an IC50 of 3.2 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 9.49 mL 47.45 mL 94.91 mL
0.5 mM 1.9 mL 9.49 mL 18.98 mL
1 mM 0.95 mL 4.75 mL 9.49 mL
5 mM 0.19 mL 0.95 mL 1.9 mL

*The above data is based on the productmolecular weight 1053.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18559
Actions Inhibitor
CAS No. 1604811-14-4
Formula C52H65ClN12O8S
M. Wt 1053.67
Purity >98%
SMILES O=C(NCCOCCOCCOCCNC(NCCCN(C)C/C=C/C(NC1=CC=C(C(NC2=CC=CC(NC3=NC=C(Cl)C(C4=CNC5=C4C=CC=C5)=N3)=C2)=O)C=C1)=O)=O)CCCC[[email protected]@H]6SC[[email protected]]([[email protected]]6([H])N7)([H])NC7=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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