Bivamelagon is a selective agonist of the melanocortin 4 receptor (MC4R) with an EC50 of 0.562 nM in a luciferase assay and 36.5 nM in a cAMP assay, demonstrating its potent activity. This compound exhibits a Ki value of 65 nM, indicating strong binding affinity to its target. Bivamelagon is valuable for research into metabolic disorders, particularly in the context of obesity and diabetes, providing insights into potential therapeutic applications.
Bivamelagon is a selective agonist of the melanocortin 4 receptor (MC4R) with an EC50 of 0.562 nM in a luciferase assay and 36.5 nM in a cAMP assay, demonstrating its potent activity. This compound exhibits a Ki value of 65 nM, indicating strong binding affinity to its target. Bivamelagon is valuable for research into metabolic disorders, particularly in the context of obesity and diabetes, providing insights into potential therapeutic applications.
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