BMS-193885

Catalog No.: A18740

neuropeptide Y1 receptor antagonist

BMS-193885

BMS-193885 Chemical Structure

CAS NO. 186185-03-5

BMS-193885 is a potent, competitive neuropeptide (NPY) Y1 antagonist (Ki = 3.3 nM, IC50 = 5.9 nM) that displays > 47, > 100, > 160, > 160 and > 160-fold selectivity over ??1, α1, Y2, Y4 and Y5 receptors respectively.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $220.00

Special Price $176.00

10 mg

Regular Price: $380.00

Special Price $304.00

50 mg

Regular Price: $980.00

Special Price $784.00

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Biological Activity

BMS-193885 is a potent, competitive neuropeptide (NPY) Y1 antagonist (Ki = 3.3 nM, IC50 = 5.9 nM) that displays > 47, > 100, > 160, > 160 and > 160-fold selectivity over ??1, α1, Y2, Y4 and Y5 receptors respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.93 mL 84.64 mL 169.29 mL
0.5 mM 3.39 mL 16.93 mL 33.86 mL
1 mM 1.69 mL 8.46 mL 16.93 mL
5 mM 0.34 mL 1.69 mL 3.39 mL

*The above data is based on the productmolecular weight 590.71. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18740
Actions Antagonist
CAS No. 186185-03-5
Formula C33H42N4O6
M. Wt 590.71
Purity >98%
Synonyms BMS193885, BMS 193885
SMILES CC1=C(C(C(=C(N1)C)C(=O)OC)c2cccc(c2)NC(=O)NCCCN3CCC(CC3)c4cccc(c4)OC)C(=O)OC
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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