BMS-470539 dihydrochloride is a selective agonist of the melanocortin-1 receptor (MC-1R), exhibiting an IC50 of 120 nM and an EC50 of 28 nM. This compound demonstrates potent anti-inflammatory properties while showing no activation of MC-3R and minimal partial agonism at MC-4R and MC-5R. BMS-470539 dihydrochloride is utilized in research focused on inflammatory conditions and the modulation of skin pigmentation.
BMS-470539 dihydrochloride is a selective agonist of the melanocortin-1 receptor (MC-1R), exhibiting an IC50 of 120 nM and an EC50 of 28 nM. This compound demonstrates potent anti-inflammatory properties while showing no activation of MC-3R and minimal partial agonism at MC-4R and MC-5R. BMS-470539 dihydrochloride is utilized in research focused on inflammatory conditions and the modulation of skin pigmentation.
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