BMS-819881

Catalog No.: A21500

MCHR1 antagonist

BMS-819881

BMS-819881 Chemical Structure

CAS NO. 1197420-05-5

BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.

Availability: In stock

Package Price Qty
1 mg
$1,184.00
5 mg
$3,551.00
10 mg
$6,049.00
50 mg
$18,147.00
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Biological Activity

BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.32 mL 106.62 mL 213.24 mL
0.5 mM 4.26 mL 21.32 mL 42.65 mL
1 mM 2.13 mL 10.66 mL 21.32 mL
5 mM 0.43 mL 2.13 mL 4.26 mL

*The above data is based on the productmolecular weight 468.95. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21500
Actions Antagonist
M. Wt 468.95
Formula C24H21ClN2O4S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1197420-05-5
Synonyms BMS 819881; BMS819881
SMILES ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[[email protected]](O)C4CC4)C=C3)C5=O)=C5S2)C=C1

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