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PDK-1 inhibitor

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Catalog No. A11148

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
BX-795 10mg A11148-10

Regular Price: $120.00

Special Price: $108.00

BX-795 25mg A11148-25

Regular Price: $250.00

Special Price: $225.00

BX-795 50mg A11148-50

Regular Price: $420.00

Special Price: $378.00

BX-795 100mg A11148-100

Regular Price: $800.00

Special Price: $720.00

BX-795 10mM * 1mL in DMSO A11148-10mM-D

Regular Price: $130.00

Special Price: $117.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

BX-795 is a potent PDK1 inhibitor that blocks PDK1/Akt signaling in tumor cells and inhibits the anchorage-dependent growth of a variety of tumor cell lines in culture or induced apoptosis.


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Publications citing Adooq Products
BX-795 Citations (1)
  • Hirosumi Tamura, .et al. Evaluation of anticancer agents using patient-derived tumor organoids characteristically similar to source tissues, Oncol Rep, 2018, Aug; 40(2): 635-646 PMID: 29917168

Chemical Information

Catalog Num A11148
Actions Inhibitor
M. Wt 591.5
Formula C23H26IN7O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 702675-74-9
Synonyms BX795

Biological Activity

BX-795 is a potent PDK1 inhibitor that blocks PDK1/Akt signaling in tumor cells and inhibits the anchorage-dependent growth of a variety of tumor cell lines in culture or induced apoptosis.
Target Value
PDK-1IC50: 6nM
c-KitIC50: 320nM
CDK2/CyclinEIC50: 430nM
Chk1IC50: 510nM
GSK-3βIC50: 620nM
PKAIC50: 840nM
KDRIC50: 1.1μM
T-FynIC50: 6.4μM
PKCIC50: 9.3μM
EGFRIC50: >10μM
Insulin ReceptorIC50: >10μM


Solubility (25°C) * In vitro DMSO 100 mg/mL (169.07 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% PEG400/0.5% Tween80/5% propylene glycol 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.91 mL 84.53 mL 169.06mL
0.5 mM 3.38 mL 16.91 mL 33.81 mL
1 mM 1.69 mL 8.45 mL 16.91 mL
5 mM 0.34 mL 1.69 mL 3.38 mL

*The above data is based on the productmolecular weight 591.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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