Fig. 1 · Structure
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CAY10669
PCAF Inhibitor
CAY10669 is a PCAF inhibitor that functions through the inhibition of histone acetyltransferase activity. With an IC50 value of 662 μM, CAY10669 enhances SAHA-induced acetylation in HEPG2 cells and promotes transgene expression in CHO-K1 cells. Additionally, it demonstrates cytotoxic effects in zebrafish embryos, making it a valuable tool for studying histone modification and gene expression regulation in various biological contexts.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1243583-88-1 |
| Applications | PCAF Inhibitor |
| Formula | C20H22O4 |
| Molecular Weight | 326.39 |
| SMILES | OC1=CC=CC(/C=C\C2=CC=C(C=C2)OCCCCC)=C1C(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.