Fig. 1 · Structure
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CCK antagonist 1
CCK Antagonist
CCK Antagonist 1 is a potent antagonist of cholecystokinin (CCK) receptors, exhibiting IC50 values of 1.1 μM for CCK1 and 4 μM for CCK2. This compound is valuable for research into the roles of CCK in cancer and mental health disorders, facilitating the exploration of therapeutic interventions targeting these pathways. Its specificity and efficacy make it a useful tool for studying the biological functions of CCK receptors.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 742116-45-6 |
| Applications | CCK Antagonist |
| Formula | C22H22N4O2 |
| Molecular Weight | 374.44 |
| SMILES | O=C(CCC1=CNC2=C1C=CC=C2)NC3=C(C)N(C)N(C4=CC=CC=C4)C3=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.