CI-988

Name: CI-988
Brand: Adooq Bioscience
SKU: A59701
Rating: 5 (288 reviews)

Catalog No.: A59701

CCK2R Antagonist

CI-988 is a potent and selective antagonist of the cholecystokinin 2 receptor (CCK2R), exhibiting an IC50 of 1.7 nM in mouse cortex assays. Demonstrating over 1600-fold selectivity for CCK2 over the CCK1 receptor, CI-988 has been shown to possess anxiolytic and anti-tumor properties. This compound is valuable for research into therapeutic applications in anxiety disorders and cancer treatment.

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Size	Price	Stock
5mg	$485.00	In stock
10mg	$800.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	CI-988 is a potent and selective antagonist of the cholecystokinin 2 receptor (CCK2R), exhibiting an IC50 of 1.7 nM in mouse cortex assays. Demonstrating over 1600-fold selectivity for CCK2 over the CCK1 receptor, CI-988 has been shown to possess anxiolytic and anti-tumor properties. This compound is valuable for research into therapeutic applications in anxiety disorders and cancer treatment.

Product Information

Catalog Num	A59701
Formula	C35H42N4O6
Molecular Weight	614.73
CAS Number	130332-27-3
SMILES	OC(CCC(N[C@H](C1=CC=CC=C1)CNC([C@](CC2=CNC3=C2C=CC=C3)(C)NC(OC4[C@H]5C[C@H](C6)C[C@@H]4C[C@H]6C5)=O)=O)=O)=O
Synonyms	PD134308

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