CMPD101

Name: CMPD101
Brand: Adooq Bioscience
SKU: A19795
Rating: 5 (288 reviews)

Catalog No.: A19795

GRK2/GRK3 inhibitor

CMPD101, is a novel membrane-permeable, small-molecule inhibitor of both GRK2 and GRK3 with IC50s of 18 nM and 5.4 nM. CMPD101 also inhibits ROCK-2 and PKCα (IC50s=1.4 μM and 8.1 μM, respectively).

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Grouped product items
Size	Price	Stock
1mg	$45.00	In stock
5mg	$105.00	In stock
10mg	$175.00	In stock
25mg	$400.00	In stock
50mg	$605.00	In stock
100mg	$915.00	In stock
*10mM 1mL in DMSO**	$125.00	In stock
Bulk Size	Bulk Discount

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Adooq Products cited in reputable paper

Biological Activity

Description

Targets

Target	Value

Product Information

Catalog Num	A19795
Formula	C24H21F3N6O
Molecular Weight	466.46
CAS Number	865608-11-3
SMILES	O=C(C1=CC(NCC2=NN=C(C3=CC=NC=C3)N2C)=CC=C1)NCC4=CC=CC=C4C(F)(F)F
Synonyms	CMPD 101, CMPD-101
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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