Biological Activity
Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 27.14 mL | 135.68 mL | 271.36 mL |
0.5 mM | 5.43 mL | 27.14 mL | 54.27 mL |
1 mM | 2.71 mL | 13.57 mL | 27.14 mL |
5 mM | 0.54 mL | 2.71 mL | 5.43 mL |
*The above data is based on the productmolecular weight 368.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21152 |
---|---|
Actions | Agonist |
M. Wt | 368.51 |
Formula | C23H32N2O2 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 165377-43-5 |
Synonyms | SA4503, SA 4503, SA-4503; AGY 94806, AGY94806, AGY-94806 |
SMILES | COC1=CC=C(CCN2CCN(CCCC3=CC=CC=C3)CC2)C=C1OC |
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