Cutamesine

Catalog No.: A21152

sigma 1 receptor agonist

Cutamesine

Cutamesine Chemical Structure

CAS NO. 165377-43-5

Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor.

Availability: In stock

Package Price Qty
10 mg
$129.00
25 mg
$257.00
50 mg
$443.00
100 mg
$758.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.14 mL 135.68 mL 271.36 mL
0.5 mM 5.43 mL 27.14 mL 54.27 mL
1 mM 2.71 mL 13.57 mL 27.14 mL
5 mM 0.54 mL 2.71 mL 5.43 mL

*The above data is based on the productmolecular weight 368.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21152
Actions Agonist
CAS No. 165377-43-5
Formula C23H32N2O2
M. Wt 368.51
Purity >98%
Synonyms SA4503, SA 4503, SA-4503; AGY 94806, AGY94806, AGY-94806
SMILES COC1=CC=C(CCN2CCN(CCCC3=CC=CC=C3)CC2)C=C1OC
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Cutamesine | Cutamesine Supplier | purchase | cost | manufacturer | order | distributor | buy 165377-43-5| 165377-43-5 Supplier | purchase 165377-43-5 | 165377-43-5 cost | 165377-43-5 manufacturer | order 165377-43-5 | 165377-43-5 distributor
Rewards