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D-Trp2,7,9 Substance P

Catalog No.: A62028
Tachykinin Antagonist
[D-Trp2,7,9] Substance P is a tachykinin antagonist primarily targeting neurokinin receptors. It exhibits Ki values of 1 μM, 1.3 μM, and approximately 9 μM for NK-1, NK-2, and NK-3 receptors, respectively. This compound is utilized in research applications focused on modulating pain, inflammation, and neurogenic responses. Its ability to selectively block neurokinin receptor activity makes it a valuable tool for exploring tachykinin-related biological processes.
[D-Trp2,7,9] Substance P 100930-11-8 Tachykinin Antagonist
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
Description[D-Trp2,7,9] Substance P is a tachykinin antagonist primarily targeting neurokinin receptors. It exhibits Ki values of 1 μM, 1.3 μM, and approximately 9 μM for NK-1, NK-2, and NK-3 receptors, respectively. This compound is utilized in research applications focused on modulating pain, inflammation, and neurogenic responses. Its ability to selectively block neurokinin receptor activity makes it a valuable tool for exploring tachykinin-related biological processes.
Product Information
Catalog NumA62028
FormulaC80H109N21O13S
Molecular Weight1604.92
CAS Number100930-11-8
Sequence shorteningRWKPQQWFWLM-NH2
SMILESCSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)CCCNC(N)=N)C(N)=O
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GPCR/G Protein > Neurokinin Receptors