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D-Trp2,7,9 Substance P

Tachykinin Antagonist

[D-Trp2,7,9] Substance P is a tachykinin antagonist primarily targeting neurokinin receptors. It exhibits Ki values of 1 μM, 1.3 μM, and approximately 9 μM for NK-1, NK-2, and NK-3 receptors, respectively. This compound is utilized in research applications focused on modulating pain, inflammation, and neurogenic responses. Its ability to selectively block neurokinin receptor activity makes it a valuable tool for exploring tachykinin-related biological processes.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	100930-11-8
Applications	Tachykinin Antagonist
Formula	C₈₀H₁₀₉N₂₁O₁₃S
Molecular Weight	1604.92
SMILES	CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)CCCNC(N)=N)C(N)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.