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Delequamine

Catalog No.: A58819
α2-Adrenergic Receptor Antagonist
Delequamine is a selective α2-adrenergic receptor antagonist with a pKi of 9.5 for α2-adrenoceptors in the rat cortex. It exhibits over 1000-fold selectivity against 5-HT1A receptors and α1-adrenoceptors. This compound is valuable for researching erectile dysfunction and exploring therapeutic options targeting adrenergic signaling pathways.
Delequamine 119905-05-4 α2-Adrenergic Receptor Antagonist
Grouped product items
Size Price Stock Qty
1mg
$205.00
In stock
5mg
$530.00
In stock
10mg
$770.00
In stock
25mg
$1,160.00
In stock
50mg
$1,525.00
In stock
100mg
$1,990.00
In stock
500mg
$3,845.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionDelequamine is a selective α2-adrenergic receptor antagonist with a pKi of 9.5 for α2-adrenoceptors in the rat cortex. It exhibits over 1000-fold selectivity against 5-HT1A receptors and α1-adrenoceptors. This compound is valuable for researching erectile dysfunction and exploring therapeutic options targeting adrenergic signaling pathways.
Product Information
Catalog NumA58819
FormulaC18H26N2O3S
Molecular Weight350.48
CAS Number119905-05-4
SMILESCS(=O)(N1[C@@]2([H])C[C@@]3([H])C4=CC=C(OC)C=C4CCN3C[C@@]2([H])CCC1)=O
SynonymsRS-15385-197
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GPCR/G Protein > Adrenergic Receptors