Desvenlafaxine-d6 is a deuterium-labeled derivative of Desvenlafaxine, which acts as a selective serotonin (5-HT) and norepinephrine reuptake inhibitor. It exhibits significant potency with IC50 values of 47.3 nM for the human serotonin transporter (hSERT) and 531.3 nM for the human norepinephrine transporter (hNET). Additionally, Desvenlafaxine shows minimal binding affinity at the human dopamine transporter, indicating its focused mechanism of action. This stable isotope is valuable for pharmacokinetic studies and metabolic profiling in neuropharmacology research.
Desvenlafaxine-d6 is a deuterium-labeled derivative of Desvenlafaxine, which acts as a selective serotonin (5-HT) and norepinephrine reuptake inhibitor. It exhibits significant potency with IC50 values of 47.3 nM for the human serotonin transporter (hSERT) and 531.3 nM for the human norepinephrine transporter (hNET). Additionally, Desvenlafaxine shows minimal binding affinity at the human dopamine transporter, indicating its focused mechanism of action. This stable isotope is valuable for pharmacokinetic studies and metabolic profiling in neuropharmacology research.
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