DMX-5804

Catalog No.: A20199

MAP4K4 inhibitor

DMX-5804

DMX-5804 Chemical Structure

CAS NO. 2306178-56-1

DMX-5804 is a potent, orally active and selective MAP4K4 inhibitor, with an IC50 of 3 nM, a pIC50 of 8.55 for human MAP4K4, less potent on MINK1/MAP4K6 (pIC50, 8.18), and TNIK/MAP4K7 (pIC50, 7.96).

Availability: In stock

Package Price Qty
5 mg
$320.00
10 mg
$500.00
50 mg
$1,500.00
100 mg
$2,500.00
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Biological Activity

DMX-5804 is a potent, orally active and selective MAP4K4 inhibitor, with an IC50 of 3 nM, a pIC50 of 8.55 for human MAP4K4, less potent on MINK1/MAP4K6 (pIC50, 8.18), and TNIK/MAP4K7 (pIC50, 7.96).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.67 mL 138.35 mL 276.71 mL
0.5 mM 5.53 mL 27.67 mL 55.34 mL
1 mM 2.77 mL 13.84 mL 27.67 mL
5 mM 0.55 mL 2.77 mL 5.53 mL

*The above data is based on the productmolecular weight 361.39. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20199
Actions Inhibitor
M. Wt 361.39
Formula C21H19N3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2306178-56-1
Synonyms DMX5804, DMX 5804
SMILES O=C1NC=NC2=C1C(C3=CC=C(OCCOC)C=C3)=CN2C4=CC=CC=C4

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