DPM-1001

Catalog No.: A18674

PTP1B inhibitor

DPM-1001

DPM-1001 Chemical Structure

CAS NO. 1471172-27-6

DPM-1001 is a potent, specific, orally bioavailable and non-competitive inhibitor of protein-tyrosine phosphatase (PTP1B) with an IC50 of 100 nM, an an analog of the specific PTP1B inhibitor trodusquemine (MSI-1436; IC50=600 nM). DPM-1001 has anti-diabetic property.

Availability: In stock

Package Price Qty
1 mg
$140.00
5 mg
$420.00
10 mg
$720.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

DPM-1001 is a potent, specific, orally bioavailable and non-competitive inhibitor of protein-tyrosine phosphatase (PTP1B) with an IC50 of 100 nM, an an analog of the specific PTP1B inhibitor trodusquemine (MSI-1436; IC50=600 nM). DPM-1001 has anti-diabetic property.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.61 mL 88.05 mL 176.1 mL
0.5 mM 3.52 mL 17.61 mL 35.22 mL
1 mM 1.76 mL 8.81 mL 17.61 mL
5 mM 0.35 mL 1.76 mL 3.52 mL

*The above data is based on the productmolecular weight 567.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18674
Actions Inhibitor
M. Wt 567.85
Formula C35H57N3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1471172-27-6
Synonyms DPM-1001; DPM1001; DPM 1001
SMILES O[[email protected]]1[[email protected]]2([H])[[email protected]@](CC[[email protected]@]3(C)[[email protected]@]2([H])CC[[email protected]]3([H])[[email protected]](C)CCC(OC)=O)([H])[[email protected]]4(C)[[email protected]@](C[[email protected]](NCCCCNCC5=CC=CC=N5)CC4)([H])C1

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy DPM-1001 | DPM-1001 Supplier | purchase | cost | manufacturer | order | distributor | buy 1471172-27-6| 1471172-27-6 Supplier | purchase 1471172-27-6 | 1471172-27-6 cost | 1471172-27-6 manufacturer | order 1471172-27-6 | 1471172-27-6 distributor
Rewards