Fig. 1 · Structure
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DSP-1053 benzenesulfonate
SERT Inhibitor
DSP-1053 benzenesulfonate is a potent selective serotonin transporter (SERT) inhibitor, exhibiting a Ki value of 1.02 nM. Additionally, it demonstrates partial agonistic activity at the 5-HT1A receptor with a Ki of 5.05 nM. Due to its profile, DSP-1053 holds potential for investigation in antidepressant efficacy and research related to serotonergic modulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1176326-78-5 |
| Applications | SERT Inhibitor |
| Formula | C32H38BrNO7S |
| Molecular Weight | 660.62 |
| SMILES | O=C1CCOC2=CC=C(CCN3CCC(CC4=CC=C(Br)C(OCCOC)=C4)CC3)C=C12.O=S(C5=CC=CC=C5)(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.