Fig. 1 · Structure
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Elismetrep
Cat. No.
A68726
CAS
1400699-64-0
TRPM8 Antagonist
Elismetrep (MT-8554) is a selective TRPM8 antagonist that inhibits the activity of the transient receptor potential melastatin 8 channel. It is shown to reduce the frequency of vasomotor symptoms and is valuable for research in pain modulation and sensory perception. Elismetrep offers potential applications in the study of disorders related to thermal sensation and nociception.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1400699-64-0 |
| Applications | TRPM8 Antagonist |
| Formula | C27H21F3N2O5S |
| Molecular Weight | 542.53 |
| Synonyms | MT-8554 |
| SMILES | O=C(C1=CC=C(S(=O)(N(CC2=CC=C(C=C2)OC(F)(F)F)C3=C(C4CC4)C5=CC=CC=C5C=N3)=O)C=C1)O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.