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Elsulfavirine sodium

VM1500A Prodrug

Elsulfavirine sodium is a prodrug that serves as an allosteric inhibitor of HIV-1 non-nucleoside reverse transcriptase, primarily through its active metabolite VM1500A. It also inhibits human carbonic anhydrase isoforms and blocks interactions between adenylosuccinate lyase and insulin-induced gene proteins, leading to decreased lipid synthesis and cancer cell proliferation. This compound demonstrates potential in HIV-1 replication inhibition and exhibits a synergistic anti-tumor effect when combined with Lenvatinib. Elsulfavirine sodium is relevant for research focusing on HIV infection and liver cancer.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	867365-40-0
Applications	VM1500A Prodrug
Formula	C₂₄H₁₇BrCl₂FN₃NaO₅S
Molecular Weight	652.27
Synonyms	R-1206 sodium
SMILES	N#CC1=CC(Cl)=CC(OC2=C(F)C(CC(NC3=CC=C(S(=O)(NC(CC)=O)=O)C=C3Cl)=O)=CC=C2Br)=C1.[Na]

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.