Fig. 1 · Structure
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EP4 receptor agonist 2
EP4 Receptor Agonist
EP4 Receptor Agonist 2 is a potent agonist of the EP4 receptor, exhibiting an EC50 value of 0.8 nM. This compound has demonstrated selectivity with Ki values of >100,000, 38,000, and 3.1 nM for the EP2, EP3, and EP4 receptors, respectively. It is a valuable tool for studying the role of EP4 signaling in various biological processes and exploring potential therapeutic applications in inflammatory and cardiovascular diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 493035-81-7 |
| Applications | EP4 Receptor Agonist |
| Formula | C27H32ClNO4 |
| Molecular Weight | 470.00 |
| SMILES | CC1=C(C=CC(Cl)=C1)C2=CC(C(O)/C=C/[C@@H]3N(C(CC3)=O)CCCCCCC(O)=O)=CC=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.