Fig. 1 · Structure
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Epaminurad hydrochloride
URAT1 Inhibitor
Epaminurad hydrochloride is a potent and selective inhibitor of URAT1 (urate transporter 1), with a Ki value of 0.057 μM. This compound exhibits partial inhibition of OAT1 and OAT3 (organic anion transporters) and acts as a uricosuric agent. Epaminurad hydrochloride is primarily utilized in research focused on gout and hyperuricemia, advancing the understanding of uric acid regulation in these conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1198153-46-6 |
| Applications | URAT1 Inhibitor |
| Formula | C14H11Br2ClN2O3 |
| Molecular Weight | 450.51 |
| Synonyms | UR-1102 hydrochloride; URC-102 hydrochloride |
| SMILES | O=C(N1C2=C(OCC1)C=CN=C2)C3=CC(Br)=C(C(Br)=C3)O.[H]Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.