Epertinib

Catalog No.: A13777

EGFR/HER2/HER4 inhibitor

Epertinib

Epertinib Chemical Structure

CAS NO. 908305-13-5

Epertinib is a potent, oral, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4, with IC50s of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib shows potent antitumor activity.

Availability: In stock

Package Price Qty
5 mg
$288.00
10 mg
$496.00
50 mg
$1,472.00
100 mg
$2,944.00
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Biological Activity

Epertinib is a potent, oral, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4, with IC50s of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib shows potent antitumor activity.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.86 mL 89.28 mL 178.57 mL
0.5 mM 3.57 mL 17.86 mL 35.71 mL
1 mM 1.79 mL 8.93 mL 17.86 mL
5 mM 0.36 mL 1.79 mL 3.57 mL

*The above data is based on the productmolecular weight 560.02. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13777
Actions Inhibitor
M. Wt 560.02
Formula C30H27ClFN5O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 908305-13-5
Synonyms S-22611, S22611, S 22611
SMILES CC#C/C(C1=CC2=C(NC3=CC=C(OCC4=CC=CC(F)=C4)C(Cl)=C3)N=CN=C2C=C1)=N\OC[[email protected]@H]5NCCOC5

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