Biological Activity
EPZ031686 is a noncompetitive inhibitor for SMYD3 and MEKK2 with a Ki=1.2 and 1.1 nM respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 16.92 mL | 84.59 mL | 169.18 mL |
0.5 mM | 3.38 mL | 16.92 mL | 33.84 mL |
1 mM | 1.69 mL | 8.46 mL | 16.92 mL |
5 mM | 0.34 mL | 1.69 mL | 3.38 mL |
*The above data is based on the productmolecular weight 591.09. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A16375 |
---|---|
Actions | Inhibitor |
CAS No. | 1808011-22-4 |
Formula | C26H34ClF3N4O4S |
M. Wt | 591.09 |
Purity | >98% |
Synonyms | EPZ-031686, EPZ 031686 |
SMILES | ClC1=CC(N2)=C(CC2=O)C=C1C(N[[email protected]@]3([H])C[[email protected]@](N4S(CC(CC5)CCN5CCCC(F)(F)F)(=O)=O)([H])CC[[email protected]@]4([H])C3)=O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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