Fig. 1 · Structure
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ER-819762
EP4 Receptor Antagonist
ER-819762 is a selective antagonist of the prostaglandin E2 (PGE2) EP4 receptor, demonstrating an EC50 value of 70 nM in human EP4 receptor assays. This compound is primarily employed in research related to rheumatoid arthritis, making it a valuable tool for investigating the role of EP4 signaling in inflammatory processes and potential therapeutic interventions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1155773-15-1 |
| Applications | EP4 Receptor Antagonist |
| Formula | C30H39N3O3 |
| Molecular Weight | 489.65 |
| SMILES | CCN1C2(CCN(CC2)CC3=CC(C)=CC(C)=C3)C(N(CC4=CC(OC)=C5)C1=O)=C[C@H](C)C4=C5OC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.