ERK5-IN-1

Catalog No.: A16232

ERK5 inhibitor

ERK5-IN-1

ERK5-IN-1 Chemical Structure

CAS NO. 1234479-76-5

ERK5-IN-1 exhibits potent inhibition of ERK5 with cellular EC50 values of 0.19 uM and enzymatic IC50 values of 0.087 uM and of LRRK2[G2019S] with enzymatic IC50 values of 0.026uM.

Availability: In stock

Package Price Qty
5 mg
$320.00
10 mg
$480.00
50 mg
$1,400.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

ERK5-IN-1 exhibits potent inhibition of ERK5 with cellular EC50 values of 0.19 uM and enzymatic IC50 values of 0.087 uM and of LRRK2[G2019S] with enzymatic IC50 values of 0.026uM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.76 mL 108.8 mL 217.61 mL
0.5 mM 4.35 mL 21.76 mL 43.52 mL
1 mM 2.18 mL 10.88 mL 21.76 mL
5 mM 0.44 mL 2.18 mL 4.35 mL

*The above data is based on the productmolecular weight 459.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A16232
Actions Inhibitor
M. Wt 459.54
Formula C25H29N7O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1234479-76-5
Synonyms ERK5 IN 1, ERK5IN1
SMILES O=C1N(C)C2=CN=C(NC3=CC=C(N4CCN(C)CC4)C=C3OC)N=C2N(C)C5=CC=CC=C15

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