ESI-05

Name: ESI-05
Brand: Adooq Bioscience
SKU: A18644
Rating: 5 (1 reviews)

Catalog No.: A18644

EPAC2 antagonist

Adooq's ESI-05 has been cited by 1 publications

ESI-05 (NSC 116966) is a specific antagonist of EPAC2 (exchange protein directly activated by cAMP 2), with an IC50 of 0.4 ?M. ESI-05 (NSC 116966) inhibits cAMP-mediated activation of EPAC2 as well as EAPC2 mediated Rap1 activation.

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Grouped product items
Size	Price	Stock
2mg	$25.00	In stock
5mg	$45.00	In stock
10mg	$85.00	In stock
25mg	$160.00	In stock
50mg	$275.00	In stock
100mg	$475.00	In stock
*10mM 1mL in DMSO**	$50.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Adooq Products cited in reputable paper

Adooq's ESI-05 has been cited by 1 publications

Yuri A Blednov, .et al. , Neuropharmacology, 2024, Jun 13:257:110035 PMID: 38876310

Biological Activity

Description	ESI-05 (NSC 116966) is a specific antagonist of EPAC2 (exchange protein directly activated by cAMP 2), with an IC50 of 0.4 ?M. ESI-05 (NSC 116966) inhibits cAMP-mediated activation of EPAC2 as well as EAPC2 mediated Rap1 activation.

Product Information

Catalog Num	A18644
Formula	C16H18O2S
Molecular Weight	274.37
CAS Number	5184-64-5
SMILES	O=S(C1=C(C)C=C(C)C=C1C)(C2=CC=C(C)C=C2)=O
Synonyms	ESI05, ESI 05
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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