Fig. 1 · Structure
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Eticlopride
D2 Receptor Antagonist
Eticlopride is a selective antagonist of the dopamine D2 receptor, demonstrating a high binding affinity for dopamine D2 as well as for α1-adrenergic, α2-adrenergic, 5HT1, and 5HT2 receptors, with Kis of 0.09, 112, 699, 6220, and 830 nM, respectively. This compound is primarily utilized in research related to antipsychotic drug development and elucidation of dopamine's role in neuropsychiatric disorders. Its pharmacological profile supports investigations into dopamine receptor modulation and its implications in various neurological conditions.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 84226-12-0 |
| Applications | D2 Receptor Antagonist |
| Formula | C17H25ClN2O3 |
| Molecular Weight | 340.85 |
| Synonyms | FLB-131 |
| SMILES | O=C(C1=C(C(CC)=CC(Cl)=C1OC)O)NC[C@H]2N(CCC2)CC |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.