Fosnetupitant

Catalog No.: A62005
Prodrug Of Netupitant
Fosnetupitant is a prodrug of Netupitant, functioning primarily as a selective antagonist of the human neurokinin-1 (NK1) receptor. With a pKi of 9.5, it offers significant inhibitory activity, making it a valuable tool in research focused on neurokinin signaling pathways. Fosnetupitant is utilized in studies related to pain management, nausea, and the effects of substance P in various biological systems.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Biological Activity
DescriptionFosnetupitant is a prodrug of Netupitant, functioning primarily as a selective antagonist of the human neurokinin-1 (NK1) receptor. With a pKi of 9.5, it offers significant inhibitory activity, making it a valuable tool in research focused on neurokinin signaling pathways. Fosnetupitant is utilized in studies related to pain management, nausea, and the effects of substance P in various biological systems.
Product Information
Catalog NumA62005
FormulaC31H35F6N4O5P
Molecular Weight688.60
CAS Number1703748-89-3
SMILESO=P(OC[N+]1(C)CCN(C2=NC=C(N(C)C(C(C)(C3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3)C)=O)C(C4=CC=CC=C4C)=C2)CC1)([O-])O
SynonymsPronetupitant
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