Fosnetupitant is a prodrug of Netupitant, functioning primarily as a selective antagonist of the human neurokinin-1 (NK1) receptor. With a pKi of 9.5, it offers significant inhibitory activity, making it a valuable tool in research focused on neurokinin signaling pathways. Fosnetupitant is utilized in studies related to pain management, nausea, and the effects of substance P in various biological systems.
Fosnetupitant is a prodrug of Netupitant, functioning primarily as a selective antagonist of the human neurokinin-1 (NK1) receptor. With a pKi of 9.5, it offers significant inhibitory activity, making it a valuable tool in research focused on neurokinin signaling pathways. Fosnetupitant is utilized in studies related to pain management, nausea, and the effects of substance P in various biological systems.
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