GDC-0810 (Brilanestrant)

Catalog No.: A15958

Estrogen receptor degrader

GDC-0810 (Brilanestrant)

GDC-0810 (Brilanestrant) Chemical Structure

CAS NO. 1365888-06-7

GDC-0810 an orally bioavailable Selective Estrogen Receptor Degrader (SERD) that demonstrates robust activity in tamoxifen-resistant breast cancer xenografts.

Availability: In stock

Package Price Qty
5 mg
$130.00
10 mg
$195.00
25 mg
$380.00
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Biological Activity

GDC-0810 an orally bioavailable Selective Estrogen Receptor Degrader (SERD) that demonstrates robust activity in tamoxifen-resistant breast cancer xenografts.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.38 mL 111.88 mL 223.76 mL
0.5 mM 4.48 mL 22.38 mL 44.75 mL
1 mM 2.24 mL 11.19 mL 22.38 mL
5 mM 0.45 mL 2.24 mL 4.48 mL

*The above data is based on the productmolecular weight 446.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15958
Actions Degrader
M. Wt 446.91
Formula C26H20ClFN2O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1365888-06-7
Synonyms RG6046, ARN-810, ARN810, ARN 810
SMILES O=C(O)/C=C/C1=CC=C(C=C1)/C(C2=CC3=C(NN=C3)C=C2)=C(CC)\C4=CC=C(C=C4Cl)F

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