Customer Appreciation Sale.
15% off with promo code "APPRECIATION2023" on check out or purchase order

GK921

Catalog No.: A21785

transglutaminase 2 (TGase) inhibitor

GK921

GK921 Chemical Structure

CAS NO. 1025015-40-0

GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.

Availability: In stock

Package Price Qty
5 mg
$135.00
10 mg
$233.00
50 mg
$690.00
100 mg
$1,380.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.
In vitro DMSO 31 mg/mL (90 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.04 mL 145.18 mL 290.35 mL
0.5 mM 5.81 mL 29.04 mL 58.07 mL
1 mM 2.9 mL 14.52 mL 29.04 mL
5 mM 0.58 mL 2.9 mL 5.81 mL

*The above data is based on the productmolecular weight 344.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21785
Actions Inhibitor
CAS No. 1025015-40-0
Formula C21H20N4O
M. Wt 344.41
Purity >98%
Synonyms GK 921, GK-921
SMILES C12=NC=CC=C1N=C(OCCN3CCCC3)C(C#CC4=CC=CC=C4)=N2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GK921 | GK921 Supplier | purchase | cost | manufacturer | order | distributor | buy 1025015-40-0| 1025015-40-0 Supplier | purchase 1025015-40-0 | 1025015-40-0 cost | 1025015-40-0 manufacturer | order 1025015-40-0 | 1025015-40-0 distributor
Rewards