GK921

Catalog No.: A21785

transglutaminase 2 (TGase) inhibitor

GK921

GK921 Chemical Structure

CAS NO. 1025015-40-0

GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.

Availability: In stock

Package Price Qty
5 mg
$135.00
10 mg
$233.00
50 mg
$690.00
100 mg
$1,380.00
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Biological Activity

GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.
In vitro DMSO 31 mg/mL (90 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.04 mL 145.18 mL 290.35 mL
0.5 mM 5.81 mL 29.04 mL 58.07 mL
1 mM 2.9 mL 14.52 mL 29.04 mL
5 mM 0.58 mL 2.9 mL 5.81 mL

*The above data is based on the productmolecular weight 344.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21785
Actions Inhibitor
CAS No. 1025015-40-0
Formula C21H20N4O
M. Wt 344.41
Solubility DMSO
Purity >98%
Synonyms GK 921, GK-921
SMILES C12=NC=CC=C1N=C(OCCN3CCCC3)C(C#CC4=CC=CC=C4)=N2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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