GLPG2451

Catalog No.: A18919

CFTR potentiator

GLPG2451

GLPG2451 Chemical Structure

CAS NO. 2055015-61-5

GLPG2451 is a cystic fibrosis transmembrane conductance regulator (CFTR) potentiator, which effectively potentiates low temperature rescued F508del CFTR with an EC50 of 11.1 nM.

Availability: In stock

Package Price Qty
5 mg
$320.00
10 mg
$520.00
50 mg
$1,500.00
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Biological Activity

GLPG2451 is a cystic fibrosis transmembrane conductance regulator (CFTR) potentiator, which effectively potentiates low temperature rescued F508del CFTR with an EC50 of 11.1 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.84 mL 119.22 mL 238.45 mL
0.5 mM 4.77 mL 23.84 mL 47.69 mL
1 mM 2.38 mL 11.92 mL 23.84 mL
5 mM 0.48 mL 2.38 mL 4.77 mL

*The above data is based on the productmolecular weight 419.38. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18919
Actions Potentiator
M. Wt 419.38
Formula C16H16F3N3O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2055015-61-5
Synonyms GLPG 2451, GLPG-2451
SMILES O=S(C1=CC=C(OC(F)(F)F)C=C1)(C2=CN=C(C(NC[[email protected]@H](O)C)=O)C(N)=C2)=O

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