Fig. 1 · Structure
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Glutaminase-IN-3
Glutaminase Inhibitor
Glutaminase-IN-3 is a selective inhibitor of glutaminase 1 (GLS1), demonstrating a potent inhibitory activity with an IC50 of 0.24 μM. This compound is designed for research applications focusing on metabolic processes and cellular metabolism dysregulation often seen in cancer and other metabolic disorders. Glutaminase-IN-3 can facilitate the study of glutamine dependency in various tumor types and provide insights into therapeutic strategies targeting glutaminase.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 1439399-45-7 |
| Applications | Glutaminase Inhibitor |
| Formula | C19H19F3N6O2S |
| Molecular Weight | 452.45 |
| SMILES | O=C(CC1=CC=CC(OC(F)(F)F)=C1)NC2=NN=C(CCCCC3=NN=C(N)S3)C=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.