CCG258208 hydrochloride (GRK2-IN-1)

Name: CCG258208 hydrochloride (GRK2-IN-1)
Brand: Adooq Bioscience
SKU: A20131
Rating: 5 (288 reviews)

Catalog No.: A20131

GRKs-IN-1, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=30 nM) and GRK5 (IC50=7.1 μM). GRKs-IN-1 is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine.

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CCG258208 hydrochloride (GRK2-IN-1) 2055990-90-2

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Grouped product items
Size	Price	Stock
1mg	$315.00	In stock
5mg	$360.00	In stock
10mg	$570.00	In stock
25mg	$1,035.00	In stock
50mg	$1,725.00	In stock
100mg	$2,355.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Biological Activity

Description

Targets

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Product Information

Catalog Num	A20131
Formula	C24H25FN4O4
Molecular Weight	452.48
CAS Number	2055990-90-2
SMILES	FC1=C(C(NCC2=NNC=C2)=O)C=C([C@H]3[C@H](COC4=CC=C(OCO5)C5=C4)CNCC3)C=C1
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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