GSK-2193874

Catalog No.: A14201
TRPV4 blocker
GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
Grouped product items
Size Price Stock Qty
1mg
$30.00
In stock
2mg
$45.00
In stock
5mg
$65.00
In stock
10mg
$120.00
In stock
25mg
$250.00
In stock
50mg
$420.00
In stock
100mg
$625.00
In stock
10mM * 1mL in DMSO
$105.00
In stock
Bulk Size
Bulk Discount
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Important Notice: For research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Biological Activity
Discription GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
Cell Research
Cell Line Type Value Description References
Product Information
Catalog Num A14201
Formula C37H38BrF3N4O
Molecular Weight 691.62
CAS Number 1336960-13-4
SMILES C1CCN(CC1)C2CCN(CC2)CC3=C(N=C4C=C(C=CC4=C3C(=O)NC5(CC5)C6=CC=CC=C6)Br)C7=CC(=CC=C7)C(F)(F)F
Synonyms GSK 2193874, GSK2193874
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 95 mg/mL (137.35 mM)
Water Insoluble
Ethanol Warmed: 48 mg/mL (69.4 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.46 mL 72.29 mL 144.59 mL
0.5 mM 2.89 mL 14.46 mL 28.92 mL
1 mM 1.45 mL 7.23 mL 14.46 mL
5 mM 0.29 mL 1.45 mL 2.89 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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