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$0.00 Biological Activity
GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
| In vitro | DMSO | 95 mg/mL (137.35 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 48 mg/mL (69.4 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 14.46 mL | 72.29 mL | 144.59 mL |
| 0.5 mM | 2.89 mL | 14.46 mL | 28.92 mL |
| 1 mM | 1.45 mL | 7.23 mL | 14.46 mL |
| 5 mM | 0.29 mL | 1.45 mL | 2.89 mL |
*The above data is based on the productmolecular weight 691.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A14201 |
|---|---|
| Actions | Blocker |
| CAS No. | 1336960-13-4 |
| Formula | C37H38BrF3N4O |
| M. Wt | 691.62 |
| Solubility | DMSO |
| Purity | >98% |
| Synonyms | GSK 2193874, GSK2193874 |
| SMILES | C1CCN(CC1)C2CCN(CC2)CC3=C(N=C4C=C(C=CC4=C3C(=O)NC5(CC5)C6=CC=CC=C6)Br)C7=CC(=CC=C7)C(F)(F)F |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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