GSK-2193874

Catalog No.: A14201

TRPV4 blocker

GSK-2193874

GSK-2193874 Chemical Structure

CAS NO. 1336960-13-4

GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.

Availability: In stock

Package Price Qty
10 mg
$130.00
25 mg
$260.00
50 mg
$425.00
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Biological Activity

GSK2193874 was identified as a selective, orally active TRPV4 blocker that inhibits Ca(2+) influx through recombinant TRPV4 channels and native endothelial TRPV4 currents.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.46 mL 72.29 mL 144.59 mL
0.5 mM 2.89 mL 14.46 mL 28.92 mL
1 mM 1.45 mL 7.23 mL 14.46 mL
5 mM 0.29 mL 1.45 mL 2.89 mL

*The above data is based on the productmolecular weight 691.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14201
Actions Blocker
M. Wt 691.62
Formula C37H38BrF3N4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1336960-13-4
Synonyms GSK 2193874, GSK2193874
SMILES C1CCN(CC1)C2CCN(CC2)CC3=C(N=C4C=C(C=CC4=C3C(=O)NC5(CC5)C6=CC=CC=C6)Br)C7=CC(=CC=C7)C(F)(F)F

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