GSK 2250665A

Name: GSK 2250665A
Brand: Adooq Bioscience
SKU: A17191
Rating: 5 (288 reviews)

Catalog No.: A17191

Itk inhibitor

GSK-2250665A is a Itk inhibitor with pKi = 9.2, it Exhibits selectivity for Itk over Aurora B kinase and Btk (pIC50 values are 6.4 and 6.5, respectively) and a panel of other kinases. Inhibits IFNγ production in PBMCs.

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Grouped product items
Size	Price	Stock
5mg	$95.00	In stock
10mg	$175.00	In stock
50mg	$535.00	In stock
100mg	$915.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	GSK-2250665A is a Itk inhibitor with pKi = 9.2, it Exhibits selectivity for Itk over Aurora B kinase and Btk (pIC50 values are 6.4 and 6.5, respectively) and a panel of other kinases. Inhibits IFNγ production in PBMCs.

Product Information

Catalog Num	A17191
Formula	C26H29N5OS
Molecular Weight	459.61
CAS Number	1246030-96-5
SMILES	CCC1=CC=C(N=C(NC3=NC(N[C@H]5CC[C@H](O)CC5)=NC(CC4=CC=CC=C4)=C3)S2)C2=C1
Synonyms	GSK2250665A, GSK-2250665A
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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