GSK2798745

Name: GSK2798745
Brand: Adooq Bioscience
SKU: A20799
Rating: 5 (288 reviews)

Catalog No.: A20799

TRPV4 ion channel blocker

GSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively.

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GSK2798745 1419609-94-1 TRPV4 ion channel blocker

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Grouped product items
Size	Price	Stock
1mg	$315.00	In stock
5mg	$690.00	In stock
10mg	$1,245.00	In stock
25mg	$2,265.00	In stock
50mg	$2,975.00	In stock
100mg	$3,995.00	In stock
Bulk Size	Bulk Discount

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Research use only. We do not sell to patients.

Data Sheet SDS

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Adooq Products cited in reputable paper

Biological Activity

Description	GSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively.

Product Information

Catalog Num	A20799
Formula	C25H28N6O3
Molecular Weight	460.53
CAS Number	1419609-94-1
SMILES	N#CC1=CC=C2N=CN(C[C@](CCC3)(C)C[C@@]43CN(C5=NC=C(C(C)(O)C)N=C5)C(O4)=O)C2=C1
Synonyms	GSK-2798745; GSK 2798745
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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