GSK4028

Catalog No.: A21906

GSK4028

GSK4028 Chemical Structure

CAS NO. 2079886-19-2

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.

Availability: In stock

Package Price Qty
5 mg
$495.00
10 mg
$853.00
50 mg
$2,530.00
100 mg
$5,060.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.51 mL 132.53 mL 265.06 mL
0.5 mM 5.3 mL 26.51 mL 53.01 mL
1 mM 2.65 mL 13.25 mL 26.51 mL
5 mM 0.53 mL 2.65 mL 5.3 mL

*The above data is based on the productmolecular weight 377.28. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21906
CAS No. 2079886-19-2
Formula C17H21BrN4O
M. Wt 377.28
Solubility DMSO
Purity >98%
Synonyms GSK 4028, GSK-4028
SMILES BrC1=C(N[[email protected]]2C[[email protected]@H](C3=CC=CC=C3)CN(C)C2)C=NN(C)C1=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GSK4028 | GSK4028 Supplier | purchase | cost | manufacturer | order | distributor | buy 2079886-19-2| 2079886-19-2 Supplier | purchase 2079886-19-2 | 2079886-19-2 cost | 2079886-19-2 manufacturer | order 2079886-19-2 | 2079886-19-2 distributor
Rewards