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Serine/threonine kinase

25 Items

per page
Set Descending Direction
Catalog No.
Product Name
Application
Product Information
Product Citation
  1. A13153
    WNK-IN-11

    WNK inhibitor

    WNK-IN-11 is an allosteric With-No-Lysine (WNK) kinase inhibitor, with an IC50 of 4 nM for WNK1.
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  2. A13188
    SRPIN340

    SRPK inhibitor

    SRPIN340 is a cell-permeable isonicotinamide that acts as an ATP-competitive SRPK1-selective inhibitor (IC50 = 0.14 and 1.8 μM, respectively, against mSRPK1 and mSRPK2) with much reduced activity against 143 other kinases.
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  3. A13220
    TA-316

    Megakaryocytes/platelets inducing agent is an inducing agent for megakaryocytes and/or platelets from pluripotent stem cells, the inducing agent being useful in treating diseases involving thrombopenia.
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  4. A15922
    ML-281

    STK33 inhibitor

    ML-281 is a potent ans selective STK33 inhibitor with IC50 value of 14 nM.
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  5. A16205
    WNK463

    pan-WNK-kinase inhibitor

    WNK463 is an orally bioavailable pan-WNK-kinase inhibitor.
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  6. A17120
    SGC GAK 1

    GAK inhibitor

    SGC GAK 1 is a high affinity cyclin G associated kinase (GAK) inhibitor.
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  7. A18395
    ZT-12-037-01

    ATP-competitive STK19 inhibitor

    ZT-12-037-01 is a potent, selective, ATP-competitive STK19 inhibitor. ZT-12-037-01 effectively blocks oncogenic NRAS-driven melanocyte malignant transformation and melanoma growth in vitro and in vivo.
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  8. A18640
    SPHINX31

    Serine/arginin kinase 1 inhibitor

    SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50 = 5.9 nM).
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  9. A18656
    LP-935509

    AAK1 inhibitor

    LP-935509 is a potent inhibitor of the Adapter protein-2 Associated Kinase 1 (AAK1).
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  10. A18792
    SRPKIN-1

    SRPK1/2 inhibitor

    SRPKIN-1 is a covalent and irreversible SRPK1/2 inhibitor with IC50s of 35.6 and 98 nM, respectively. Anti-angiogenesis effect.
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  11. A19702
    BAY-524

    Bub1 inhibitor

    BAY-524 is a Bub1 inhibitor, with an IC50 of 450 nM for human Bub1 in the presence of 2 mM ATP.
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  12. A19710
    BAY-320

    Bub1 inhibitor

    BAY-320 is a Bub1 inhibitor, with an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.
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  13. A19806
    GCN2iB

    GCN2 inhibitor

    GCN2iB is an ATP-competitive inhibitor of a serine/threonine-protein kinase general control nonderepressible 2 (GCN2), with an IC50 of 2.4 nM.
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  14. A19868
    BAY-1816032

    BUB1 kinase inhibitor

    BAY-1816032 is a potent and oral available BUB1 (budding uninhibited by benzimidazoles 1) kinase inhibitor with an IC50 of 7 nM.
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  15. A19970
    2OH-BNPP1

    BUB1 kinase inhibitor

    2OH-BNPP1 is an inhibitor of BUB1 kinase, a Ser/Thr kinase, used for the treatment of cancer.
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  16. A20412
    GCN2-IN-1

    GCN2 inhibitor

    GCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase (GCN2) inhibitor with an IC50 of <0.3 μM in the enzyme assay and an IC50 of 0.3-3 μM in the cell assay.
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  17. A20447
    STK16-IN-1

    STK16 kinase inhibitor

    STK16-IN-1 is a STK16 kinase inhibitor with an IC50 of 295 nM.
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  18. A21906
    GSK4028

    GSK4027 Negative Control

    GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
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  19. A22301
    BioE-1115

    PASK inhibitor

    BioE-1115 is a highly selective and potent PAS kinase (PASK) inhibitor with an IC50 of ~4 nM. BioE-1115 is also a potent casein kinase 2α inhibitor with an IC50 of ~10 μM.
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  20. A22319
    DCLK1-IN-1

    DCLK1 domain probe

    DCLK1-IN-1 is a selective, oral bioavailability in vivo-compatible chemical probe of the doublecortin like kinase 1 (DCLK1 kinase) domain.
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  21. AP2740
    STK16 Antibody

    Serine/Threonine Kinase 16, Mouse Anti Human
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  22. AP4746
    STK16 Human

    Serine/Threonine Kinase 16 Human Recombinant
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  23. AP4747
    STK17B Human

    Serine/Threonine Kinase 17B Human Recombinant
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  24. AP4748
    STK3 Human

    Serine/Threonine Kinase 3 Human Recombinant
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  25. AP4749
    STK17A Human

    Serine/Threonine Kinase 17A Human Recombinant
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25 Items

per page
Set Descending Direction