Biological Activity
GW791343 HCl acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2) and a positive allosteric modulator of rat P2X7.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 20.67 mL | 103.35 mL | 206.7 mL |
0.5 mM | 4.13 mL | 20.67 mL | 41.34 mL |
1 mM | 2.07 mL | 10.33 mL | 20.67 mL |
5 mM | 0.41 mL | 2.07 mL | 4.13 mL |
*The above data is based on the productmolecular weight 483.8 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A11107 |
---|---|
Actions | Modulator |
M. Wt | 483.8 |
Formula | C20H24F2N4O.3HCl |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1019779-04-4 |
Synonyms | GW-791343 |
SMILES | CC1=C(C=C(C=C1)CN2CCNCC2)NC(=O)CNC3=CC(=C(C=C3)F)F.Cl.Cl.Cl |
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