Catalog No.: A13165

CBP/p300 bromodomain inhibitor


I-CBP112 Chemical Structure

CAS NO. 1640282-31-0

I-CBP112 is a highly potent and selective p300/CBP bromodomain inhibitor (IC50 ~0.14-0.17 uM for CBP and ~0.625 uM for p300).

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Biological Activity

I-CBP112 is a highly potent and selective p300/CBP bromodomain inhibitor (IC50 ~0.14-0.17 uM for CBP and ~0.625 uM for p300).
In vitro DMSO 86 mg/mL (183.53 mM)
Water 86 mg/mL (183.53 mM)
Ethanol 86 mg/mL (183.53 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.34 mL 106.7 mL 213.41 mL
0.5 mM 4.27 mL 21.34 mL 42.68 mL
1 mM 2.13 mL 10.67 mL 21.34 mL
5 mM 0.43 mL 2.13 mL 4.27 mL

*The above data is based on the productmolecular weight 468.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13165
Actions Inhibitor
CAS No. 1640282-31-0
Formula C27H36N2O5
M. Wt 468.59
Purity >98%
Synonyms ICBP112
SMILES CCC(=O)N1CCOC2=C(C1)C=C(C=C2OC[[email protected]]3CCCN(C3)C)C4=CC(=C(C=C4)OC)OC

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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